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Evidence for the in Vitro Bioactivation of Aminopyrazole Derivatives: Trapping Reactive Aminopyrazole Intermediates Using Glutathione Ethyl Ester in Human Liver Microsomes

  • Eileen Ryan
  • , Benjamin J. Morrow
  • , Catherine F. Hemley
  • , Jo Anne Pinson
  • , Susan A. Charman
  • , Francis C.K. Chiu
  • , Richard C. Foitzik
  • Monash University
  • Cancer Therapeutics CRC

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Pharmacology, Toxicology and Pharmaceutical Science